SCHEMBL8914335

SCHEMBL8914335

CC(C)[C@H](NS(=O)(=O)c1cccc2c(Cl)cccc12)C(=O)O.NC(=O)N1CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
HPGD P15428 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MAPK1 P28482 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
MYLK Q15746 2/20 0.44
MEN1 O00255 1/20 0.44
TP53 P04637 1/20 0.44
NFKB1 P19838 1/20 0.44
KMT2A Q03164 1/20 0.44
GMNN O75496 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8914317 0.90 CYP3A4 (0.46) ALDH1A1KDM4EHSD17B10NPSR1MAPK1
SCHEMBL8913765 0.82 F2 (0.49) MAPK1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8913812 0.81 ROCK2 (0.51) ALDH1A1KDM4EHSD17B10MAPK1CYP1A2
SCHEMBL8914340 0.81 CYP3A4 (0.47) ALDH1A1KDM4EHSD17B10HPGDCASP1
SCHEMBL8915067 0.80 MMP2 (0.56) SLC1A3SLC1A2SLC1A1MMP12MMP2
SCHEMBL8912385 0.76 KDM4E (0.48) ALDH1A1KDM4EHSD17B10HPGDCASP1
SCHEMBL8912748 0.76 MMP2 (0.63) SLC1A3SLC1A2SLC1A1MMP12MMP2
SCHEMBL8914327 0.75 CYP3A4 (0.48) ALDH1A1KDM4EHSD17B10NPSR1MAPK1
SCHEMBL8914173 0.72 MAPK1 (0.53) ALDH1A1KDM4EHSD17B10CASP1CASP7
SCHEMBL8912770 0.72 ROCK2 (0.53) ALDH1A1KDM4EHSD17B10MAPK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663174-A ANTIINFLAMMATORY AGENTS, INHIBITOR OF KINASES, ANTIARTHRITIC AGENTS PHARNO-WEDROPHARM GMBH (DE) 1997-09-02 US disclosed
EP-0602028-B1 AROMATIC SULFONAMIDE DERIVATIVES, THEIR USE AS ENZYME INHIBITORS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PHARNO WEDROPHARM GMBH (DE) 1996-01-17 EP disclosed