SCHEMBL8914575

SCHEMBL8914575

CC1=C(C(=O)OC2CCCC2)C(c2cc(F)ccc2F)C(C(=O)n2ccnc2)=C(C)N1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.49
ACHE P22303 1/20 0.40
MAPT P10636 1/20 0.39
NR3C2 P08235 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7245462 0.81 MAPT (0.60) TP53MAPT
Imidazole SCHEMBL8914572 0.78 TP53 (0.47) TP53ACHEMAPTNR3C2
SCHEMBL8096562 0.77 TP53 (0.52) TP53ACHEMAPTNR3C2
SCHEMBL8914307 0.73 TP53 (0.47) TP53ACHEMAPTNR3C2
SCHEMBL6945801 0.72 MAPT (0.50) TP53MAPT
SCHEMBL7887451 0.71 NR1I2 (0.55) TP53MAPT
SCHEMBL8912934 0.65 CYP2C9 (0.49) TP53ACHEMAPTNR3C2
SCHEMBL10729302 0.64 CYP2C9 (0.66) TP53MAPT
SCHEMBL10726831 0.64 CYP2C9 (0.66) TP53MAPT
SCHEMBL27424745 0.64 POLB (0.42) TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658934-A Aryl-substituted alkoxycarbonyl-1,4-dihydropyridine-5-carboxylic acid esters BAYER AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed