SCHEMBL8914946

SCHEMBL8914946

S=C(NCCOc1ccccc1)Nc1cccnc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL6 P41182 1/20 0.66
SMN1; SMN2 Q16637 3/20 0.58
XBP1 P17861 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
ALDH1A1 P00352 6/20 0.57
KDM4E B2RXH2 2/20 0.57
NOTUM Q6P988 1/20 0.56
LMNA P02545 2/20 0.54
RAB9A P51151 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
MAPT P10636 1/20 0.53
HTT P42858 1/20 0.53
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
HPGD P15428 1/20 0.50
MAPK1 P28482 1/20 0.50
NPC1 O15118 1/20 0.50
GAA P10253 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8914794 0.96 BCL6 (0.64) BCL6SMN1; SMN2XBP1NPSR1ALDH1A1
SCHEMBL8915611 0.92 BCL6 (0.63) BCL6SMN1; SMN2XBP1NPSR1ALDH1A1
SCHEMBL8914521 0.89 ALDH1A1 (0.57) BCL6SMN1; SMN2XBP1NPSR1ALDH1A1
SCHEMBL8915482 0.85 SMN1; SMN2 (0.62) SMN1; SMN2XBP1NPSR1ALDH1A1LMNA
SCHEMBL8915354 0.81 L3MBTL1 (0.59) SMN1; SMN2XBP1NPSR1ALDH1A1LMNA
SCHEMBL16286371 0.81 NAMPT (0.54) BCL6SMN1; SMN2ALDH1A1KDM4ERAB9A
SCHEMBL11828701 0.79 BCL6 (0.69) BCL6ALDH1A1KDM4EMAPTHPGD
Hydrochloric Acid SCHEMBL11830789 0.77 BCL6 (0.68) BCL6ALDH1A1KDM4EMAPTHPGD
SCHEMBL8915664 0.77 L3MBTL1 (0.58) SMN1; SMN2XBP1NPSR1ALDH1A1LMNA
SCHEMBL6814444 0.77 SMN1; SMN2 (0.62) SMN1; SMN2XBP1NPSR1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696140-A FOR TREATMENT OF ASTHMA, ALLERGIES, NERVOUS SYSTEM DISORDERS OR CANCER LEO PHARMACEUTICAL PRODUCTS LTD. (DK) 1997-12-09 US disclosed
US-5563160-A NERVOUS SYSTEM DISORDERS, ANTIHISTAMINE, ANTIALLERGENS Leo Pharmaceutical Products Ltd. A/S (L.o slashed.vens Kemiske Fabrik Produktionsaktieselskab) (DK) 1996-10-08 US disclosed
EP-0660823-B1 N-CYANO-N'-PYRIDYLGUANIDINES AS SEROTONIN ANTAGONISTS LEO PHARM PROD LTD (DK) 1996-08-14 EP disclosed
EP-0660823-A1 N-CYANO-N'-PYRIDYLGUANIDINES AS SEROTONIN ANTAGONISTS. LEO PHARM PROD LTD (DK) 1995-07-05 EP disclosed
WO-1994006770-A1 N-CYANO-N'-PYRIDYLGUANIDINES AS SEROTONIN ANTAGONISTS Leo Pharmaceutical Products Ltd. A/S (Løvens Kemiske Fabrik Produktionsaktieselskab) (DK) 1994-03-31 WO disclosed