SCHEMBL8915070

SCHEMBL8915070

CC(=O)N(CCCCN)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.61
NPC1 O15118 1/20 0.49
JAK2 O60674 1/20 0.49
RAB9A P51151 1/20 0.49
PAX8 Q06710 1/20 0.49
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TSHR P16473 2/20 0.46
GLA P06280 1/20 0.46
TP53 P04637 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
ACHE P22303 2/20 0.44
LTB4R2 Q9NPC1 1/20 0.42
ICMT O60725 1/20 0.42
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10460057 0.87 ADRA2C (0.53) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL607964 0.84 NPC1 (0.67) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL10099720 0.83 MEN1 (0.62) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL1208763 0.83 NPC1 (0.69) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL9809230 0.83 NPC1 (0.69) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL4574813 0.83 NPC1 (0.49) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL817611 0.82 NPC1 (0.59) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL28132503 0.81 NPC1 (0.51) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL28142261 0.81 NPC1 (0.51) ADRA2CNPC1JAK2RAB9APAX8
SCHEMBL18358943 0.81 HRH3 (0.48) ADRA2CNPC1JAK2RAB9APAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624917-A Method of inhibiting squalene synthetase TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-29 US disclosed
EP-0541037-A2 Squalene synthetase inhibitory composition and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-05-12 EP disclosed