SCHEMBL8915514

SCHEMBL8915514

Nc1ccc(CCN2CCC3(CC2)Sc2ccc(N)cc2S3)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.46
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
THPO P40225 1/20 0.40
MTOR P42345 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
HRH3 Q9Y5N1 2/20 0.36
MBTD1 Q05BQ5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912806 0.76 KCNJ1 (0.60) SIGMAR1HRH3KCNJ1KCNH2
Hydrochloric Acid SCHEMBL8920931 0.73 KCNH2 (0.44) ALDH1A1SMN1; SMN2KCNH2LMNA
SCHEMBL12281936 0.73 SIGMAR1 (0.55) SIGMAR1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL15651638 0.71 SIGMAR1 (0.53) SIGMAR1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL16670770 0.71 SIGMAR1 (0.49) SIGMAR1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5651768 0.70 SIGMAR1 (0.64) SIGMAR1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL1877934 0.70 HRH3 (0.68) SIGMAR1ALDH1A1CYP1A2CYP3A4TDP1
SCHEMBL8565829 0.70 SIGMAR1 (0.51) SIGMAR1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL28356053 0.70 SIGMAR1 (0.58) SIGMAR1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL2234644 0.70 SIGMAR1 (0.63) SIGMAR1ALDH1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed