SCHEMBL8915544

SCHEMBL8915544

O=P(O)(O)C(NCCCCCC[S+]([O-])c1ccccc1)P(=O)(O)O.[NaH].[NaH]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 5/20 0.38
CA12 O43570 3/20 0.38
S1PR2 O95136 1/20 0.37
S1PR4 O95977 1/20 0.37
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
CA14 Q9ULX7 5/20 0.35
MMP2 P08253 3/20 0.35
MMP8 P22894 3/20 0.35
MMP14 P50281 3/20 0.35
CA2 P00918 2/20 0.35
CA1 P00915 1/20 0.35
ACP3 P15309 3/20 0.33
FDPS P14324 4/20 0.33
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8915532 0.92 CA9 (0.35) CA9CA12S1PR2S1PR4S1PR1
SCHEMBL8914943 0.81 POLB (0.39) CA9CA12CA2CA1
SCHEMBL9082979 0.79 POLB (0.40) CA9CA12CA2CA1
SCHEMBL8914859 0.71 FDPS (0.50) CA9CA12FDPSHDAC3HDAC4
SCHEMBL8917287 0.71 LAP3 (0.33) S1PR2S1PR4S1PR1S1PR3HDAC3
SCHEMBL8915288 0.71 LAP3 (0.33) S1PR2S1PR4S1PR1S1PR3HDAC3
SCHEMBL17187190 0.71 S1PR2 (0.40) CA9CA12S1PR2S1PR4S1PR1
SCHEMBL8917274 0.70 FDPS (0.45) FDPSCFTR
SCHEMBL8915283 0.70 FDPS (0.45) FDPSCFTR
SCHEMBL14990095 0.70 KDM1A (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624917-A Method of inhibiting squalene synthetase TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-29 US disclosed
EP-0541037-A2 Squalene synthetase inhibitory composition and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-05-12 EP disclosed