SCHEMBL8916149

SCHEMBL8916149

c1ccc2c(c1)CCN(CCSc1ccnc(CSc3nc4ccccc4[nH]3)c1)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.50
NOS1 P29475 1/20 0.50
NOS2 P35228 1/20 0.50
CYP1A2 P05177 3/20 0.49
CYP2E1 P05181 3/20 0.49
CYP2C8 P10632 3/20 0.49
CYP2D6 P10635 3/20 0.49
CYP2C9 P11712 3/20 0.49
CYP2B6 P20813 3/20 0.49
CYP2C19 P33261 3/20 0.49
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.48
HTR1A P08908 2/20 0.48
DRD2 P14416 2/20 0.48
HTR7 P34969 2/20 0.48
DRD3 P35462 2/20 0.48
HRH1 P35367 1/20 0.48
RAB9A P51151 5/20 0.48
GRIN2A Q12879 1/20 0.43
GRIN2B Q13224 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8914916 0.80 RAB9A (0.49) NOS3NOS1NOS2CYP1A2CYP2E1
SCHEMBL8914989 0.78 KDM4E (0.61) KDM4EALDH1A1HTR1ADRD2HTR7
SCHEMBL9275286 0.77 AR (0.64) NOS3NOS1NOS2CYP1A2CYP2E1
SCHEMBL9279489 0.76 RAB9A (0.65) NOS3NOS1NOS2CYP1A2CYP2E1
SCHEMBL8923805 0.76 CYP2C9 (0.59) NOS3NOS1NOS2CYP1A2CYP2E1
SCHEMBL9279504 0.75 RAB9A (0.69) NOS3NOS1NOS2CYP1A2CYP2E1
SCHEMBL9052895 0.74 ALDH1A1 (0.45) NOS3NOS1NOS2CYP1A2CYP2E1
SCHEMBL7848521 0.72 HTR1A (0.44) NOS3NOS1NOS2CYP1A2CYP2E1
SCHEMBL8915109 0.72 RAB9A (0.43) NOS2CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL8915115 0.72 RAB9A (0.40) NOS2CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616581-A BACTERICIDES YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-04-01 US disclosed
US-5504082-A BACTERICIDE FOR HELICOBACTER, ANTIULCER AGENT, GASTRIC ACIDSUPPRESSOR YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-04-02 US disclosed
EP-0644191-A1 PYRIDINE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-22 EP disclosed