SCHEMBL8916299

SCHEMBL8916299

O=C1c2cccc(F)c2C(=O)c2c(F)cccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.54
MAPK1 P28482 5/20 0.54
ALDH1A1 P00352 4/20 0.54
TDP1 Q9NUW8 4/20 0.54
MAOA P21397 2/20 0.54
LMNA P02545 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TSHR P16473 2/20 0.54
HPGD P15428 1/20 0.54
ALOX15 P16050 1/20 0.54
MAOB P27338 1/20 0.54
HTT P42858 1/20 0.54
HSD17B10 Q99714 1/20 0.54
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
CDC25B P30305 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5866470 0.92 CA1 (0.52) MAPTMAPK1ALDH1A1TDP1MAOA
SCHEMBL10716838 0.92 MAOA (0.52) MAPTMAPK1ALDH1A1TDP1MAOA
SCHEMBL760904 0.91 ADORA2A (0.57) MAPTMAPK1ALDH1A1TDP1MAOA
SCHEMBL13487412 0.87 CA1 (0.52) MAPTMAPK1ALDH1A1TDP1MAOA
SCHEMBL8669578 0.86 MEN1 (0.55) MAPTMAPK1ALDH1A1TDP1MAOA
SCHEMBL31307459 0.85 CA1 (0.43) MAPTMAPK1ALDH1A1TDP1MAOA
SCHEMBL7805629 0.82 CA1 (0.44) MAPTMAPK1ALDH1A1TDP1MAOA
SCHEMBL2072999 0.81 MAPT (0.52) MAPTMAPK1ALDH1A1TDP1MAOA
SCHEMBL13487411 0.81 PTPRC (0.59) MAPTMAPK1ALDH1A1MAOALMNA
SCHEMBL13487410 0.81 PTPRC (0.57) MAPTMAPK1ALDH1A1TDP1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 52 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691442-A RADIATION TRANSPARENT POLYMERS WITH PHENOL ENDCAPPING THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1997-11-25 US disclosed
EP-0180042-B1 METAL PLATED POLY(ARYL ETHER) CONTAINING ARTICLES AMOCO CORPORATION (US) 1992-11-11 EP disclosed
US-5064929-A Tough, transparent optical films MOBAY CORPORATION (US) 1991-11-12 US disclosed
US-4841009-A Substantially linear monomeric composition and liquid crystal polymeric compositions derived therefrom AMOCO CORPORATION (US) 1989-06-20 US disclosed
US-4820790-A HEAT RESISTANCE, SOLVENT RESISTANCE AMOCO CORPORATION (US) 1989-04-11 US disclosed
EP-0168539-B1 BLENDS COMPRISING COPOLYMERS OF POLYPHENYLENE OXIDES AND POLY(ARYL ETHER)S, STYRENE POLYMERS AND/OR COPOLYMERS, POLY(ARYL ETHER)S AND/OR POLYPHENYLENE OXIDES AMOCO CORPORATION (US) 1989-03-29 EP disclosed
US-H521-H Thermosetting polysulfones SOLVAY ADVANCED POLYMERS, LLC 1988-09-06 US disclosed
US-4767838-A HIGH TEMPERATURE AND SOLVENT RESISTANT; HYDROQUINONE WITH A DIHALO OR DINITRO-BENZOPHENONE AND OTHER AROMATIC COMPOUND AMOCO CORPORATION (US) 1988-08-30 US disclosed
EP-0111327-B1 A COMPOSITION USEFUL FOR MAKING CIRCUIT BOARD SUBSTRATES AMOCO CORPORATION (US) 1988-06-29 EP disclosed
US-4687833-A HYDROQUINONE, 4,4'-DIHALO OR DINITRO KETONE, BASE, APROTIC SOLVENT AMOCO CORPORATION (US) 1987-08-18 US disclosed
US-4240974-A 1,2,3,4,9,9-HEXAHALO-1,4-DIHYDRO-1,4-METHANO-NAPHTHALENE-5,8 -DISULFONATE LITTLE JULIAN R (US) 1980-12-23 US disclosed
US-4232142-A Production of polyarylene ether sulphones and ketones IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1980-11-04 US disclosed
US-4175175-A POLYSULFONES, POLYSULFONAMIDES UNION CARBIDE CORPORATION (US) 1979-11-20 US disclosed
US-4174457-A Carbamate UNIROYAL, INC. (US) 1979-11-13 US disclosed
US-4108837-A THERMOPLASTIC, REACTING DIALKALI METAL SALT OF A DIHYDRIC PHENOL WITH A SUBSTITUTED DIHALOBENZENOID IN PRESENCE OF A SOLVENT UNION CARBIDE CORPORATION (US) 1978-08-22 US disclosed
US-4080408-A FIRE RETARDANTS UNIROYAL, INC. (US) 1978-03-21 US disclosed
US-4058568-A FIRE RETARDANT UNIROYAL, INC. (US) 1977-11-15 US disclosed
US-4051109-A POLYETHERSULFONES IMPERIAL CHEMICAL INDUSTRIES LIMITED (EN) 1977-09-27 US disclosed
US-4009200-A FIREPROOFING POLYMERS UNIROYAL, INC. (US) 1977-02-22 US disclosed
US-3949002-A POLYMER AND PHARMACEUTICAL INTERMEDIATE IMPERIAL CHEMICAL INDUSTRIES LIMITED (EN) 1976-04-06 US disclosed