SCHEMBL8917168

SCHEMBL8917168

Cc1cccc2c(N3CC[N]CC3)coc12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.44
ADRB1 P08588 2/20 0.34
KDM4E B2RXH2 4/20 0.33
GAA P10253 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
MAPT P10636 1/20 0.33
ALDH1A1 P00352 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
PHGDH O43175 1/20 0.32
HTR6 P50406 1/20 0.32
POLB P06746 1/20 0.32
HPGD P15428 1/20 0.32
CES1 P23141 1/20 0.32
NCF1 P14598 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2A6 P11509 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917181 0.82 HTR6 (0.34) PRKDCKDM4EMAPTALDH1A1PHGDH
SCHEMBL8918038 0.76 ADORA2A (0.37) PRKDCADRB1KDM4EL3MBTL1MAPT
SCHEMBL1447600 0.72 ADRB1 (0.62) ADRB1KDM4EGAAL3MBTL1MAPT
SCHEMBL217611 0.71 ADRB1 (0.60) ADRB1ALDH1A1HPGD
SCHEMBL8917845 0.71 KCNA3 (0.36) KDM4ECES1CYP1A2CYP2A6
SCHEMBL8917269 0.70 ADRB1 (0.34) PRKDCADRB1KDM4EGAAL3MBTL1
SCHEMBL8917934 0.70 MAPT (0.39) PRKDCKDM4EMAPTALDH1A1PHGDH
SCHEMBL8917729 0.70 PRKDC (0.45) PRKDCKDM4EMAPTALDH1A1PHGDH
SCHEMBL1448499 0.69 KDM4E (0.51) KDM4EGAAL3MBTL1MAPTALDH1A1
SCHEMBL2607400 0.68 CYP2A6 (0.48) MAPTALDH1A1TDP1POLBCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US claimed
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed