SCHEMBL8917269

SCHEMBL8917269

Cc1cccc2c(N3CC[N]CC3)csc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.34
MAPT P10636 3/20 0.34
TP53 P04637 3/20 0.34
KDM4E B2RXH2 3/20 0.33
GAA P10253 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
LMNA P02545 1/20 0.33
PRKDC P78527 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HTR6 P50406 1/20 0.32
LPAR2 Q9HBW0 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 2/20 0.31
CYP2A6 P11509 1/20 0.31
CYP3A4 P08684 1/20 0.31
HTR1A P08908 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916972 0.82 MAPT (0.33) MAPTTP53KDM4EL3MBTL1LMNA
SCHEMBL8920541 0.76 ADRB1 (0.34) ADRB1MAPTTP53KDM4ELMNA
SCHEMBL1447600 0.72 ADRB1 (0.62) ADRB1MAPTKDM4EGAAL3MBTL1
SCHEMBL217611 0.71 ADRB1 (0.60) ADRB1LMNAHTTRECQLSMN1; SMN2
SCHEMBL8917168 0.70 PRKDC (0.44) ADRB1MAPTKDM4EGAAL3MBTL1
SCHEMBL8917044 0.70 MAPT (0.48) MAPTTP53LMNARECQLALDH1A1
SCHEMBL8918997 0.70 DRD2 (0.35) CYP1A2CYP2A6
SCHEMBL8919052 0.70 MAPT (0.58) MAPTTP53LMNARECQLALDH1A1
SCHEMBL1448499 0.69 KDM4E (0.51) MAPTKDM4EGAAL3MBTL1LMNA
SCHEMBL8404365 0.68 CYP1A2 (0.48) MAPTGAACYP1A2CYP2A6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed