SCHEMBL8917255

SCHEMBL8917255

CCC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.76
KDM4E B2RXH2 4/20 0.76
TDP1 Q9NUW8 3/20 0.76
HTT P42858 1/20 0.76
KMT2A Q03164 7/20 0.71
MEN1 O00255 6/20 0.71
POLB P06746 3/20 0.71
MAPT P10636 3/20 0.71
LMNA P02545 4/20 0.67
TSHR P16473 2/20 0.65
CYP3A4 P08684 2/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
ABCB11 O95342 1/20 0.65
CYP1A2 P05177 1/20 0.65
ADRA2A P08913 1/20 0.65
CYP2D6 P10635 1/20 0.65
CHRM1 P11229 1/20 0.65
TBXA2R P21731 1/20 0.65
SLC6A2 P23975 1/20 0.65
SLC6A4 P31645 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8914869 0.90 ALDH1A1 (0.72) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL7933991 0.87 ALDH1A1 (0.72) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL3142795 0.87 ALDH1A1 (0.72) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL1064531 0.86 ALDH1A1 (0.71) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL27663681 0.86 ALDH1A1 (0.70) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL8913178 0.86 ALDH1A1 (0.71) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL8917304 0.85 ALDH1A1 (0.69) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL2853078 0.85 KMT2A (0.70) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL9987888 0.85 ALDH1A1 (0.69) ALDH1A1KDM4ETDP1HTTKMT2A
SCHEMBL13417633 0.84 ALDH1A1 (0.76) ALDH1A1KDM4ETDP1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1993339-B Aromatic compound OTSUKA PHARMA CO LTD 2013-05-22 CN disclosed
US-20120238750-A1 AROMATIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. 2012-09-20 US disclosed
US-20120238750-A1 AROMATIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. 2012-09-20 US disclosed
US-8236826-B2 Diarylether derivatives as antitumor agents OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2012-08-07 US disclosed
US-8236826-B2 Diarylether derivatives as antitumor agents OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2012-08-07 US disclosed
US-8188277-B2 Aromatic compounds for suppressing the generation of collagen OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2012-05-29 US disclosed
US-8188277-B2 Aromatic compounds for suppressing the generation of collagen OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2012-05-29 US disclosed
US-20100004438-A1 DIARYLETHER DERIVATIVES AS ANTITUMOR AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2010-01-07 US disclosed
US-20100004438-A1 DIARYLETHER DERIVATIVES AS ANTITUMOR AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2010-01-07 US disclosed
CN-101321529-A Diaryl aether derivant as antineoplastic agent OTSUKA PHARMA CO LTD (JP) 2008-12-10 CN disclosed
US-20070270422-A1 Aromatic Compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-11-22 US disclosed
US-20070270422-A1 Aromatic Compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-11-22 US disclosed
CN-1993339-A Aromatic compound OTSUKA PHARMA CO LTD (JP) 2007-07-04 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120238750-A1 AROMATIC COMPOUND CBR1, CBR3, CYP1A1 ALDH1A1 565/4885KDM4E 1219/4885TDP1 4207/4885
US-20100004438-A1 DIARYLETHER DERIVATIVES AS ANTITUMOR AGENTS ROS1, CBR1, CBR3 ALDH1A1 265/4885KDM4E 2010/4885TDP1 3760/4885
US-20070270422-A1 Aromatic Compounds COL1A1, COL2A1, COL14A1 ALDH1A1 475/4885KDM4E 988/4885TDP1 3705/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.