SCHEMBL8917343

SCHEMBL8917343

CS(=O)(=O)c1ccc(-n2nc(C(F)F)c3ccc4cc(OC(F)(F)F)ccc4c32)cc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.41
EPHX2 P34913 1/20 0.40
PTGS1 P23219 2/20 0.38
CYP2C9 P11712 1/20 0.38
NPY5R Q15761 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
GRIA2 P42262 1/20 0.35
NR3C1 P04150 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918829 0.89 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL8919647 0.85 CYP1A2 (0.46) PTGS2EPHX2PTGS1CYP2C9CYP1A2
SCHEMBL8917301 0.84 PTGS2 (0.45) PTGS2PTGS1CYP2C9
SCHEMBL8916673 0.83 PTGS2 (0.44) PTGS2PTGS1CYP2C9
SCHEMBL8916712 0.82 PTGS2 (0.41) PTGS2PTGS1CYP2C9
SCHEMBL8919630 0.82 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL8917466 0.82 PTGS2 (0.41) PTGS2PTGS1CYP2C9
SCHEMBL8919075 0.81 PTGS2 (0.40) PTGS2PTGS1CYP2C9
SCHEMBL8917535 0.81 LCK (0.40) PTGS2PTGS1
SCHEMBL8921429 0.80 PTGS2 (0.42) PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed
WO-1996009293-A1 BENZ[g]INDAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO disclosed