SCHEMBL8918829

SCHEMBL8918829

COc1ccc2c(ccc3c(C(F)F)nn(-c4ccc(S(C)(=O)=O)cc4)c32)c1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.43
PTGS1 P23219 7/20 0.43
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
KMT2A Q03164 1/20 0.39
TEK Q02763 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9232444 0.90 PTGS2 (0.54) PTGS2PTGS1CA1CA2CA9
SCHEMBL8917343 0.89 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL8917301 0.86 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL8916673 0.85 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL8919630 0.84 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL8917466 0.84 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL8916712 0.84 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL8919075 0.83 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL8917535 0.83 LCK (0.40) PTGS2PTGS1CA1CA2CA9
SCHEMBL8921429 0.83 PTGS2 (0.42) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed