SCHEMBL8917391

SCHEMBL8917391

C=CCc1cccnc1NN1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
ACHE P22303 2/20 0.44
DTYMK P23919 1/20 0.44
GPR119 Q8TDV5 6/20 0.42
F13A1 P00488 3/20 0.40
TGM2 P21980 3/20 0.40
TGM1 P22735 3/20 0.40
KDR P35968 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CKS1B P61024 1/20 0.38
SKP1 P63208 1/20 0.38
SKP2 Q13309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8985778 0.82 POLB (0.50) POLBACHEDTYMKGPR119CKS1B
SCHEMBL20818668 0.73 POLB (0.50) POLBACHEDTYMKGPR119MEN1
SCHEMBL30476354 0.73 POLB (0.50) POLBACHEDTYMKGPR119MEN1
SCHEMBL7402298 0.72 ALDH1A1 (0.52) POLBACHEDTYMKGPR119ALDH1A1
SCHEMBL30476397 0.71 POLB (0.50) POLBACHEDTYMKGPR119MEN1
SCHEMBL20818148 0.71 POLB (0.50) POLBACHEDTYMKGPR119MEN1
SCHEMBL8923840 0.71 ACHE (0.48) POLBACHEDTYMKGPR119MEN1
SCHEMBL31652019 0.71 POLB (0.55) POLBACHEDTYMKGPR119CKS1B
SCHEMBL11366665 0.70 POLB (0.54) POLBACHEDTYMKGPR119CKS1B
SCHEMBL21358044 0.70 KDM4E (0.39) MEN1ALDH1A1LMNAKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686610-A Pyridyl piperazine compound PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
US-5599930-A Substituted indoles as anti-AIDS pharmaceuticals THE UPJOHN COMPANY (US) 1997-02-04 US disclosed
WO-1993001181-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS THE UPJOHN COMPANY (US) 1993-01-21 WO disclosed