SCHEMBL8985778

SCHEMBL8985778

C=CCc1cccnc1N1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
GPR119 Q8TDV5 7/20 0.46
ACHE P22303 2/20 0.46
DTYMK P23919 1/20 0.46
KIT P10721 2/20 0.46
GBA1 P04062 1/20 0.46
TRPV1 Q8NER1 2/20 0.45
TRPA1 O75762 2/20 0.45
CKS1B P61024 1/20 0.44
SKP1 P63208 1/20 0.44
SKP2 Q13309 1/20 0.44
PDE10A Q9Y233 1/20 0.43
RBP4 P02753 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31652019 0.87 POLB (0.55) POLBGPR119ACHEDTYMKKIT
SCHEMBL11366665 0.86 POLB (0.54) POLBGPR119ACHEDTYMKKIT
SCHEMBL5901303 0.85 POLB (0.53) POLBGPR119ACHEDTYMKKIT
SCHEMBL8923840 0.82 ACHE (0.48) POLBGPR119ACHEDTYMKKIT
SCHEMBL8917391 0.82 POLB (0.47) POLBGPR119ACHEDTYMKCKS1B
SCHEMBL3287405 0.81 PDE10A (0.51) POLBGPR119ACHEDTYMKKIT
SCHEMBL31046329 0.80 POLB (0.57) POLBGPR119ACHEDTYMKKIT
SCHEMBL3436722 0.80 POLB (0.57) POLBGPR119ACHEDTYMKKIT
SCHEMBL2715768 0.80 POLB (0.57) POLBGPR119ACHEDTYMKKIT
SCHEMBL6469181 0.79 POLB (0.57) POLBGPR119ACHEDTYMKKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563142-A INHIBITORS OF VIRAL REVERSE TRANSCRIPTASE THE UPJOHN COMPANY (US) 1996-10-08 US disclosed
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP disclosed
US-5489593-A Anti-aids piperazines THE UPJOHN COMPANY (US) 1996-02-06 US disclosed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO disclosed