SCHEMBL8917578

SCHEMBL8917578

O=C(CF)NC1NCCNC1c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 7/20 0.39
MAPT P10636 1/20 0.39
POLB P06746 2/20 0.38
MDM2 Q00987 1/20 0.37
GAA P10253 2/20 0.37
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36
HSD17B10 Q99714 2/20 0.36
GRM5 P41594 1/20 0.35
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918459 0.83 ALDH1A1 (0.36) ALDH1A1KMT2AKDM4EPOLBMDM2
SCHEMBL8919141 0.78 CTH (0.31) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL8916129 0.76 MDM2 (0.34) ALDH1A1KMT2AKDM4EMAPTMDM2
SCHEMBL8917001 0.73 KDM4E (0.33) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL8917889 0.73 CTH (0.34) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL8916767 0.72 KDM5A (0.34) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL8916653 0.72 SLC2A1 (0.36) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL20840557 0.68 SLC1A2 (0.40) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL27793415 0.67 NISCH (0.40) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL27793412 0.67 DDB1 (0.37) ALDH1A1KMT2AKDM4EMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686610-A Pyridyl piperazine compound PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed