SCHEMBL8917595

SCHEMBL8917595

CC(C)Nc1cnnc(Cl)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 1/20 0.46
AOC1 P19801 3/20 0.36
AOC3 Q16853 2/20 0.36
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GAA P10253 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NR4A2 P43354 1/20 0.32
PDE10A Q9Y233 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8791827 0.74 LRRK2 (0.32) KAT2BPDE10A
SCHEMBL23341540 0.72
SCHEMBL8406855 0.72 LRRK2 (0.35) KAT2BGABRA1GABRG2GABRB3GABRA5
SCHEMBL18227477 0.72 AOC1 (0.36) AOC1AOC3GABRA1GABRG2GABRB3
SCHEMBL30557610 0.72 AOC1 (0.36) AOC1AOC3GABRA1GABRG2GABRB3
SCHEMBL8923769 0.69 KAT2B (0.47) KAT2BAOC1AOC3GAATDP1
SCHEMBL11831985 0.65 TDP1 (0.40) KAT2BAOC1AOC3GAATDP1
SCHEMBL19841858 0.64 IDO1 (0.43) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL30867766 0.64
SCHEMBL17200370 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686610-A Pyridyl piperazine compound PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
US-5563142-A INHIBITORS OF VIRAL REVERSE TRANSCRIPTASE THE UPJOHN COMPANY (US) 1996-10-08 US disclosed
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP disclosed
US-5489593-A Anti-aids piperazines THE UPJOHN COMPANY (US) 1996-02-06 US disclosed
WO-1993001181-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS THE UPJOHN COMPANY (US) 1993-01-21 WO disclosed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO disclosed