SCHEMBL8918036

SCHEMBL8918036

CN(C)CC(=O)c1cc2c(s1)CCCC(=O)N2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
TSHR P16473 1/20 0.50
RAB9A P51151 1/20 0.50
DAO P14920 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
MCL1 Q07820 1/20 0.33
ALDH1A1 P00352 6/20 0.33
MAPT P10636 1/20 0.32
ABL1 P00519 1/20 0.32
RIN1 Q13671 1/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 1/20 0.32
POLB P06746 2/20 0.31
PKM P14618 1/20 0.31
CRBN Q96SW2 1/20 0.31
CYP3A4 P08684 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916424 0.86 MEN1 (0.47) CYP2C19MEN1KMT2ATSHRRAB9A
SCHEMBL8915783 0.73 CDC7 (0.36) CYP2C19MEN1KMT2ADAOL3MBTL1
SCHEMBL8915779 0.70 RAB9A (0.93) CYP2C19MEN1KMT2ATSHRRAB9A
SCHEMBL26983413 0.68 KDM4E (0.46) CYP2C19MEN1KMT2ATSHRRAB9A
SCHEMBL19228585 0.67 RAB9A (0.60) CYP2C19MEN1KMT2ATSHRRAB9A
SCHEMBL8917940 0.65 MEN1 (0.53) CYP2C19MEN1KMT2ATSHRRAB9A
SCHEMBL31411868 0.60 HPGD (0.47) CYP2C19MEN1KMT2ATSHRRAB9A
SCHEMBL18538442 0.60 GSK3B (0.31)
Bicarbonate SCHEMBL28617859 0.59 CRBN (0.77) CYP2C19MEN1KMT2ATSHRRAB9A
Bicarbonate SCHEMBL28617862 0.59 CRBN (0.77) CYP2C19MEN1KMT2ATSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed
EP-0596125-A1 CONDENSED THIOPHENE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed