SCHEMBL8918356

SCHEMBL8918356

COC(=O)c1c(C)nc(N)c(C#N)c1-c1cccc([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
HPGD P15428 2/20 0.49
GAA P10253 1/20 0.49
ACHE P22303 2/20 0.47
CACNB4 O00305 1/20 0.47
CACNA1A O00555 1/20 0.47
CACNA1G O43497 1/20 0.47
CACNG3 O60359 1/20 0.47
CACNA1F O60840 1/20 0.47
CACNA1H O95180 1/20 0.47
BCHE P06276 1/20 0.47
CACNB3 P54284 1/20 0.47
CACNA2D1 P54289 1/20 0.47
CACNG7 P62955 1/20 0.47
CACNA1B Q00975 1/20 0.47
CACNA1D Q01668 1/20 0.47
CACNB1 Q02641 1/20 0.47
CACNG1 Q06432 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10746185 0.85 ALDH1A1 (0.70) ALDH1A1MEN1KMT2AHPGDGAA
SCHEMBL6137255 0.81 SMN1; SMN2 (0.56) ALDH1A1MEN1KMT2AHPGDGAA
SCHEMBL9452419 0.81 ALDH1A1 (0.56) ALDH1A1MEN1KMT2AGAAACHE
SCHEMBL4384277 0.81 ALDH1A1 (0.64) ALDH1A1MEN1KMT2AHPGDGAA
SCHEMBL6956520 0.81 ALDH1A1 (0.64) ALDH1A1MEN1KMT2AHPGDGAA
SCHEMBL7887160 0.80 MEN1 (0.53) ALDH1A1MEN1KMT2AACHECACNB4
SCHEMBL10745416 0.79 ALDH1A1 (0.54) ALDH1A1MEN1KMT2AHPGDGAA
SCHEMBL6956135 0.79 SMN1; SMN2 (0.62) ALDH1A1MEN1KMT2AHPGDGAA
SCHEMBL10747824 0.78 ACHE (0.47) ALDH1A1MEN1KMT2AHPGDGAA
SCHEMBL8917637 0.78 CACNB4 (0.54) ALDH1A1KMT2AHPGDGAACACNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670525-A Substituted 4-phenyl-6-amino-nicotinic acid compounds useful in the treatment of CNS disorders BAYER AKTIENGESELLSCHAFT (DE) 1997-09-23 US disclosed
EP-0705820-A1 6-Amino-nicotinic acid derivatives and their use as selective K-channel modulators BAYER AG (DE) 1996-04-10 EP disclosed