SCHEMBL8918642

SCHEMBL8918642

C=CCn1c(=O)oc2cc(Br)cnc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
HSD17B10 Q99714 2/20 0.36
KMT2A Q03164 2/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
PDE4B Q07343 2/20 0.36
NPC1 O15118 1/20 0.36
CYP3A4 P08684 1/20 0.35
ADORA2B P29275 5/20 0.35
ADORA2A P29274 3/20 0.35
ADORA3 P0DMS8 2/20 0.34
ADORA1 P30542 1/20 0.34
USP2 O75604 1/20 0.33
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17418888 0.80 PDE4B (0.43) ALDH1A1HSD17B10KMT2APDE4BNPC1
SCHEMBL23198637 0.79 HSD17B10 (0.38) ALDH1A1HSD17B10KMT2APDE4B
SCHEMBL8627148 0.77 PDE4B (0.36) ALDH1A1HSD17B10KMT2APDE4BNPC1
SCHEMBL8918139 0.74 HSD17B10 (0.38) ALDH1A1HSD17B10KMT2ACASP1CASP7
SCHEMBL7316292 0.74 NPC1 (0.63) ALDH1A1HSD17B10NPC1LMNAHPGD
SCHEMBL7328412 0.73 HSD17B10 (0.53) ALDH1A1HSD17B10KMT2APDE4BNPC1
SCHEMBL8626898 0.72 TSHR (0.56) ALDH1A1HSD17B10KMT2ACASP1CASP7
SCHEMBL32686762 0.71 PDE4B (0.38) ALDH1A1HSD17B10KMT2APDE4BNPC1
SCHEMBL8919804 0.71 LMNA (0.42) ALDH1A1HSD17B10KMT2APDE4BNPC1
SCHEMBL23198630 0.70 IDO1 (0.38) ALDH1A1HSD17B10KMT2APDE4BNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed