SCHEMBL8627148

SCHEMBL8627148

N#CCn1c(=O)oc2cc(Br)cnc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.36
HSD17B10 Q99714 1/20 0.36
NPC1 O15118 1/20 0.36
ADORA2B P29275 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
GFER P55789 1/20 0.33
KMT2A Q03164 1/20 0.33
KMO O15229 2/20 0.32
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32
PGR P06401 1/20 0.32
PDE4A P27815 1/20 0.32
ADORA2A P29274 1/20 0.32
PDE4C Q08493 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918139 0.86 HSD17B10 (0.38) PDE4BHSD17B10NPC1ALDH1A1HPGD
SCHEMBL17418888 0.80 PDE4B (0.43) PDE4BHSD17B10NPC1ALDH1A1LMNA
SCHEMBL8624599 0.80 ADORA2B (0.35) PDE4BADORA2BALDH1A1KMOKDM4E
SCHEMBL8918642 0.77 ALDH1A1 (0.36) PDE4BHSD17B10NPC1ADORA2BALDH1A1
SCHEMBL7316292 0.74 NPC1 (0.63) HSD17B10NPC1ALDH1A1LMNAHPGD
SCHEMBL7328412 0.73 HSD17B10 (0.53) PDE4BHSD17B10NPC1ALDH1A1LMNA
SCHEMBL8626898 0.72 TSHR (0.56) HSD17B10NPC1ADORA2BALDH1A1LMNA
SCHEMBL32686762 0.71 PDE4B (0.38) PDE4BHSD17B10NPC1ALDH1A1LMNA
SCHEMBL8919804 0.71 LMNA (0.42) PDE4BHSD17B10NPC1ALDH1A1LMNA
SCHEMBL23198637 0.70 HSD17B10 (0.38) PDE4BHSD17B10ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5767128-A ANALGESICS ADIR ET COMPAGNIE (FR) 1998-06-16 US disclosed
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed