SCHEMBL8918664

SCHEMBL8918664

COc1ccc2c(ccc3c(C(F)F)nn(-c4ccc(S(C)(=O)=O)cc4)c32)c1F

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.47
PTGS1 P23219 6/20 0.41
ABCB11 O95342 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917817 0.86 PTGS2 (0.38) PTGS2PTGS1
SCHEMBL8918665 0.85 PTGS2 (0.39) PTGS2PTGS1
SCHEMBL8917393 0.82 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL8921405 0.80 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL8918829 0.79 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL9233583 0.78 PTGS2 (0.52) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8920821 0.78 PTGS2 (0.38) PTGS2PTGS1
SCHEMBL8916673 0.77 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL8917890 0.77 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL8917301 0.76 PTGS2 (0.45) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed