SCHEMBL8919214

SCHEMBL8919214

CC/C=C(C)/C=C\CNC(=O)Cc1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
GAA P10253 1/20 0.48
LMNA P02545 1/20 0.47
EPHX2 P34913 1/20 0.46
ERCC1 P07992 1/20 0.46
ERCC4 Q92889 1/20 0.46
FAAH O00519 2/20 0.45
KMT2A Q03164 2/20 0.44
PKM P14618 1/20 0.44
POLB P06746 1/20 0.44
NAPRT Q6XQN6 1/20 0.43
MAPT P10636 1/20 0.43
RECQL P46063 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918492 0.91 FAAH (0.48) CYP1A2CYP3A4CYP2C9GAALMNA
SCHEMBL8919580 0.82 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C9GAALMNA
SCHEMBL8918394 0.81 THRB (0.52) CYP1A2CYP3A4GAAKMT2AMAPT
SCHEMBL8919867 0.81 THRB (0.52) CYP1A2CYP3A4GAAKMT2AMAPT
SCHEMBL8918390 0.81 THRB (0.52) CYP1A2CYP3A4GAAKMT2AMAPT
SCHEMBL12409531 0.76 CYP1A2 (0.66) CYP1A2CYP3A4CYP2C9GAALMNA
SCHEMBL22109517 0.76 PKM (0.52) FAAHKMT2APKMPOLBMAPT
SCHEMBL13196041 0.74 CYP1A2 (0.62) CYP1A2CYP3A4CYP2C9GAALMNA
SCHEMBL10398808 0.73 TRPV1 (0.62) CYP1A2CYP3A4CYP2C9GAAEPHX2
SCHEMBL10398809 0.73 TRPV1 (0.62) CYP1A2CYP3A4CYP2C9GAAEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691366-A UNSATURATED NITRO OXIME FORMED BY REACTION OF DINITROGEN TRIOXIDE WITH DIOLEFIN ETHER, SULFIDE OR AMINE TO BE USED AS VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed