SCHEMBL8919241

SCHEMBL8919241

CC=C(C=CCNC(=O)c1ccc(NS(C)(=O)=O)nc1)CC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
CTSL P07711 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
P4HTM Q9NXG6 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HCAR3 P49019 3/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
HCAR2 Q8TDS4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919231 1.00 ALDH1A1 (0.37) ALDH1A1CTSLCTSSCTSKP4HTM
SCHEMBL8919032 0.81 KDM4E (0.51) ALDH1A1KMT2AHDAC1HDAC6MAPT
SCHEMBL8919568 0.80 HDAC1 (0.48) MEN1KMT2AHDAC1HDAC6
SCHEMBL8919561 0.80 HDAC1 (0.48) MEN1KMT2AHDAC1HDAC6
SCHEMBL8920234 0.74 THRB (0.54) ALDH1A1MEN1KMT2AHDAC3HDAC4
SCHEMBL8921545 0.74 THRB (0.54) ALDH1A1MEN1KMT2AHDAC3HDAC4
SCHEMBL8921547 0.74 THRB (0.54) ALDH1A1MEN1KMT2AHDAC3HDAC4
SCHEMBL751341 0.73 MAOB (0.47) ALDH1A1P4HTMMEN1KMT2AHCAR3
SCHEMBL8919987 0.73 SMN1; SMN2 (0.55) ALDH1A1KMT2AHDAC3HDAC1HDAC2
SCHEMBL12999502 0.72 CA1 (0.50) P4HTMKMT2AHCAR3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691366-A UNSATURATED NITRO OXIME FORMED BY REACTION OF DINITROGEN TRIOXIDE WITH DIOLEFIN ETHER, SULFIDE OR AMINE TO BE USED AS VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5623078-A Process for producing an intermediate of a new quinolone compound CHISSO CORPORATION (JP) 1997-04-22 US disclosed
US-5495023-A VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-27 US disclosed
WO-1993010097-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-27 WO disclosed