SCHEMBL8919618

SCHEMBL8919618

CCCC=C(C)C=CCNC(=O)c1cccnc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.50
KMT2A Q03164 5/20 0.48
MEN1 O00255 4/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
SREBF2 Q12772 1/20 0.47
RAB9A P51151 5/20 0.46
NPC1 O15118 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC3 O15379 1/20 0.46
HDAC2 Q92769 1/20 0.46
GAA P10253 2/20 0.45
MAPT P10636 2/20 0.44
GFER P55789 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HDAC6 Q9UBN7 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919613 1.00 THRB (0.50) THRBKMT2AMEN1CYP1A2CYP3A4
SCHEMBL8918394 0.90 THRB (0.52) THRBKMT2AMEN1CYP1A2CYP3A4
SCHEMBL8918390 0.90 THRB (0.52) THRBKMT2AMEN1CYP1A2CYP3A4
SCHEMBL8919867 0.90 THRB (0.52) THRBKMT2AMEN1CYP1A2CYP3A4
SCHEMBL8921909 0.86 THRB (0.56) THRBKMT2AMEN1CYP1A2CYP3A4
SCHEMBL8921907 0.86 THRB (0.56) THRBKMT2AMEN1CYP1A2CYP3A4
SCHEMBL8918492 0.81 FAAH (0.48) KMT2ACYP1A2CYP3A4GAAMAPT
SCHEMBL8921547 0.79 THRB (0.54) THRBKMT2AMEN1CYP1A2CYP3A4
SCHEMBL8920234 0.79 THRB (0.54) THRBKMT2AMEN1CYP1A2CYP3A4
SCHEMBL8921545 0.79 THRB (0.54) THRBKMT2AMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691366-A UNSATURATED NITRO OXIME FORMED BY REACTION OF DINITROGEN TRIOXIDE WITH DIOLEFIN ETHER, SULFIDE OR AMINE TO BE USED AS VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5495023-A VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-27 US disclosed
WO-1993010097-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-27 WO disclosed