SCHEMBL8920395

SCHEMBL8920395

CN(C[C@@H](c1ccccc1)N1CCC(O)C1)C(=O)Cc1ccc(C(F)(F)F)cc1N

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 15/20 0.54
CYP2D6 P10635 1/20 0.43
OPRK1 P41145 1/20 0.43
CCR5 P51681 1/20 0.41
POLQ O75417 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195719 1.00 TACR1 (0.54) TACR1CYP2D6OPRK1CCR5POLQ
SCHEMBL8436169 0.87 TACR1 (0.51) TACR1CYP2D6OPRK1CCR5
SCHEMBL6526246 0.82 OPRK1 (0.49) TACR1CYP2D6OPRK1
SCHEMBL7646549 0.79 OPRK1 (0.66) CYP2D6OPRK1
SCHEMBL6350906 0.79 OPRK1 (0.66) CYP2D6OPRK1
SCHEMBL7168125 0.79 OPRK1 (0.66) CYP2D6OPRK1
SCHEMBL8438187 0.76 OPRK1 (0.52) TACR1CYP2D6OPRK1CCR5
SCHEMBL8433573 0.74 SIGMAR1 (0.47) TACR1CYP2D6OPRK1CCR5
SCHEMBL6481037 0.73 OPRK1 (0.67) TACR1OPRK1CCR5
SCHEMBL8670577 0.73 CCR5 (0.54) TACR1CYP2D6OPRK1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688955-A ANALGESICS ADOLOR CORPORATION (US) 1997-11-18 US disclosed