SCHEMBL8920505

SCHEMBL8920505

CCc1c(CCN2CCC(c3coc4cc(OC)ccc34)CC2)sc2c1CCN(C(C)=O)C2

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.39
P2RX3 P56373 1/20 0.39
DRD2 P14416 6/20 0.37
MAPT P10636 4/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 2/20 0.37
KMT2A Q03164 2/20 0.37
SLC6A4 P31645 1/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
THRB P10828 1/20 0.37
MCHR1 Q99705 2/20 0.36
HTR2A P28223 5/20 0.36
DRD3 P35462 5/20 0.36
BRD3 Q15059 2/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35
DRD4 P21917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917985 0.94 CTSS (0.40) CTSSDRD2MAPTALDH1A1SLC6A4
SCHEMBL8917881 0.90 CTSS (0.40) CTSSDRD2SLC6A4MCHR1HTR2A
SCHEMBL8916768 0.90 CTSS (0.40) CTSSDRD2MAPTMEN1KMT2A
SCHEMBL8916164 0.90 CTSS (0.48) CTSSDRD2MAPTSLC6A4MCHR1
Hydrochloric Acid SCHEMBL8917167 0.90 CTSS (0.40) CTSSDRD2MAPTMEN1KMT2A
Hydrochloric Acid SCHEMBL8918060 0.89 CTSS (0.48) CTSSDRD2MAPTSLC6A4MCHR1
SCHEMBL8919111 0.88 DRD2 (0.51) DRD2SLC6A4HTR2ADRD3
SCHEMBL8916977 0.87 CTSS (0.37) CTSSDRD2MAPTSLC6A4POLB
SCHEMBL8917017 0.86 HTR2A (0.46) DRD2SLC6A4HTR2ADRD3DRD4
SCHEMBL8916989 0.86 DRD2 (0.38) CTSSDRD2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed