SCHEMBL8921130

SCHEMBL8921130

O=C(O)CCCSc1c(O)c2ccc(Cl)cc2[nH]c1=O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.50
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 2/20 0.50
GRIN2D O15399 2/20 0.48
GRIN3B O60391 2/20 0.48
GRIN1 Q05586 2/20 0.48
GRIN2A Q12879 2/20 0.48
GRIN2B Q13224 2/20 0.48
GRIN2C Q14957 2/20 0.48
GRIN3A Q8TCU5 2/20 0.48
MEN1 O00255 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
KMT2A Q03164 1/20 0.47
GPR17 Q13304 1/20 0.45
GSK3B P49841 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8920754 0.86 ALDH1A1 (0.48) ALDH1A1KDM4EGRIN2DGRIN3BGRIN1
SCHEMBL8921443 0.86 MAPT (0.67) MAPTALDH1A1KDM4EGRIN2DGRIN3B
SCHEMBL8920133 0.84 KDM4E (0.51) MAPTALDH1A1KDM4EGRIN2DGRIN3B
SCHEMBL8921390 0.84 KDM4E (0.67) ALDH1A1KDM4EGRIN2DGRIN3BGRIN1
SCHEMBL8919874 0.83 GSK3B (0.55) ALDH1A1KDM4EGRIN2DGRIN3BGRIN1
SCHEMBL8923489 0.83 KDM4E (0.50) MAPTALDH1A1KDM4EGRIN2DGRIN3B
SCHEMBL8920782 0.83 KDM4E (0.73) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL8920155 0.82 KDM4E (0.54) MAPTALDH1A1KDM4EGRIN2DGRIN3B
SCHEMBL8920123 0.78 KDM4E (0.52) MAPTALDH1A1KDM4EGRIN2DGRIN3B
SCHEMBL8921828 0.77 ALDH1A1 (0.61) MAPTALDH1A1KDM4EGRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633379-A N-METHYLASPARTIC ACID ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-05-27 US disclosed