SCHEMBL8920754

SCHEMBL8920754

COC(=O)CCCSc1c(O)c2ccc(Cl)cc2[nH]c1=O

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
EGFR P00533 1/20 0.47
GSK3B P49841 2/20 0.47
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
GRIN1 Q05586 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
GRIN2C Q14957 1/20 0.44
GRIN3A Q8TCU5 1/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
KMT2A Q03164 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8921828 0.88 ALDH1A1 (0.61) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8921130 0.86 MAPT (0.50) ALDH1A1GSK3BGRIN2DGRIN3BGRIN1
SCHEMBL8920215 0.84 KDM4E (0.63) ALDH1A1EGFRMEN1KMT2AKDM4E
SCHEMBL8919874 0.82 GSK3B (0.55) ALDH1A1GSK3BGRIN2DGRIN3BGRIN1
SCHEMBL8921390 0.80 KDM4E (0.67) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8925163 0.79 ALDH1A1 (0.62) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8921245 0.78 GRIN2D (0.49) ALDH1A1GSK3BGRIN2DGRIN3BGRIN1
SCHEMBL8920133 0.78 KDM4E (0.51) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8921443 0.78 MAPT (0.67) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8923489 0.77 KDM4E (0.50) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633379-A N-METHYLASPARTIC ACID ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-05-27 US claimed
US-5633379-A N-METHYLASPARTIC ACID ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-05-27 US disclosed