SCHEMBL8923406

SCHEMBL8923406

CC(C)(C)OC(=O)N1CC[C@@H](S(C)(=O)=O)C[C@]1(O)Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 1/20 0.44
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
NR1H2 P55055 3/20 0.39
NR1H3 Q13133 3/20 0.39
GPR119 Q8TDV5 3/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
PTPRB P23467 1/20 0.38
PTPN11 Q06124 1/20 0.38
KDM4E B2RXH2 1/20 0.38
PKM P14618 1/20 0.38
TGFBR1 P36897 1/20 0.38
GRIN2B Q13224 2/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8923491 0.85 STS (0.43) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL8923498 0.85 STS (0.43) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL1843456 0.77
SCHEMBL28638548 0.75 STS (0.43) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL28632434 0.73 STS (0.42) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL2951728 0.69 OPRD1 (0.53) STSGPR119KDM4EPKM
SCHEMBL20137861 0.69 STS (0.68) STSGPR119JAK2JAK1PTPRB
SCHEMBL9937601 0.69 STS (0.46) STSGPR119JAK2JAK1KDM4E
SCHEMBL16080215 0.68 JAK2 (0.40) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL6535958 0.68 MEN1 (0.41) STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5646144-A FOR TREATING DISORDERS IN WHICH SUBSTANCE P PLAYS A PART IN DEVELOPMENT CIBA-GEIGY CORPORATION (US) 1997-07-08 US disclosed
US-5541195-A SUBSTANCE P ANTAGONISTS CIBA-GEIGY CORPORATION (US) 1996-07-30 US disclosed
US-5310743-A Substance P antagonist CIBA-GEIGY CORP. (US) 1994-05-10 US disclosed