SCHEMBL8923498

SCHEMBL8923498

CC(C)(C)OC(=O)N1CC[C@@H](OS(C)(=O)=O)C[C@]1(O)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
STS P08842 1/20 0.43
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
NR1H2 P55055 3/20 0.38
NR1H3 Q13133 3/20 0.38
KLK7 P49862 1/20 0.37
GPR119 Q8TDV5 3/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
PTPRB P23467 1/20 0.37
PTPN11 Q06124 1/20 0.37
HCRTR2 O43614 1/20 0.37
TGFBR1 P36897 1/20 0.36
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8923491 1.00 STS (0.43) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL28638548 0.88 STS (0.43) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL8923406 0.85 STS (0.44) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL1843456 0.76
SCHEMBL28632434 0.75 STS (0.42) STSPDE4APDE4BPDE4CPDE4D
SCHEMBL21410627 0.75 GPR119 (0.37) NR1H2NR1H3GPR119
SCHEMBL22533463 0.74 GPR119 (0.37) GPR119
SCHEMBL9200786 0.73 NR1H2 (0.54) STSNR1H2NR1H3KLK7GPR119
SCHEMBL9200782 0.73 NR1H2 (0.54) STSNR1H2NR1H3KLK7GPR119
SCHEMBL28566941 0.73 STS (0.38) STSNR1H2NR1H3KLK7GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5646144-A FOR TREATING DISORDERS IN WHICH SUBSTANCE P PLAYS A PART IN DEVELOPMENT CIBA-GEIGY CORPORATION (US) 1997-07-08 US disclosed
US-5541195-A SUBSTANCE P ANTAGONISTS CIBA-GEIGY CORPORATION (US) 1996-07-30 US disclosed
US-5310743-A Substance P antagonist CIBA-GEIGY CORP. (US) 1994-05-10 US disclosed