SCHEMBL8923758

SCHEMBL8923758

CN(C(N)=O)C(=O)CCSC[C@@H]1C[C@H](O[Si](C)(C)C(C)(C)C)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 1/20 0.34
CCR5 P51681 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8694615 1.00 ALDH1A1 (0.34) ALDH1A1MAPTHPGDCCR5NPC1
SCHEMBL8692334 0.93 CCR5 (0.35) ALDH1A1MAPTHPGDCCR5NPC1
SCHEMBL8925236 0.91 CCR5 (0.35) ALDH1A1MAPTHPGDCCR5TDP1
SCHEMBL8694603 0.91 CCR5 (0.35) ALDH1A1MAPTHPGDCCR5TDP1
SCHEMBL8924545 0.89 CCR5 (0.34) ALDH1A1MAPTHPGDCCR5TDP1
SCHEMBL8696188 0.89 ALDH1A1 (0.36) ALDH1A1MAPTHPGDCCR5NPC1
SCHEMBL8921898 0.89 ALDH1A1 (0.36) ALDH1A1MAPTHPGDCCR5NPC1
SCHEMBL8694952 0.88 MAPT (0.36) ALDH1A1MAPTHPGDRAB9AL3MBTL1
SCHEMBL8924296 0.88 MAPT (0.36) ALDH1A1MAPTHPGDRAB9AL3MBTL1
SCHEMBL9520885 0.87 ALDH1A1 (0.37) ALDH1A1MAPTHPGDCCR5NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5641770-A THIENAMYCINS ANTIBIOTICS CHONG KUN DANG CORP. (KR) 1997-06-24 US disclosed
EP-0674640-A1 2-(2-SUBSTITUTED PYRROLIDIN-4-YL)THIO-CARBAPENEM DERIVATIVES CHONG KUN DANG CORP (KR) 1995-10-04 EP disclosed
WO-1994014811-A1 2-(2-SUBSTITUTED PYRROLIDIN-4-YL)THIO-CARBAPENEM DERIVATIVES CHONG KUN DANG CORP. (KR) 1994-07-07 WO disclosed