SCHEMBL8924065

SCHEMBL8924065

CCOC(=O)COP(=O)(CN[C@@H](Cc1ccc(-c2ccccc2)cc1OC)c1nnn[nH]1)OCC(=O)OCC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.36
ADRB3 P13945 4/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MME P08473 2/20 0.34
ECE1 P42892 1/20 0.34
AGTR2 P50052 1/20 0.34
ROCK2 O75116 4/20 0.34
ROCK1 Q13464 4/20 0.34
KDR P35968 3/20 0.33
EGFR P00533 2/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
DYRK3 O43781 1/20 0.33
MAP4K4 O95819 1/20 0.33
CDK1 P06493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8924096 1.00 ADRB1 (0.36) ADRB1ADRB3KDM4EALDH1A1TP53
SCHEMBL8922872 0.87 MME (0.46) KDM4EALDH1A1TP53MAPTHPGD
SCHEMBL8922845 0.87 MME (0.46) KDM4EALDH1A1TP53MAPTHPGD
SCHEMBL8923691 0.85 ROCK2 (0.36) ADRB1ADRB3MMEECE1AGTR2
SCHEMBL8923716 0.85 ROCK2 (0.36) ADRB1ADRB3MMEECE1AGTR2
SCHEMBL8924880 0.84 KDM4E (0.38) KDM4EALDH1A1MAPTHPGDHSD17B10
SCHEMBL8924951 0.84 KDM4E (0.38) KDM4EALDH1A1MAPTHPGDHSD17B10
SCHEMBL8920285 0.84 ECE1 (0.46) ADRB1ADRB3MMEECE1AGTR2
SCHEMBL8920227 0.84 ECE1 (0.46) ADRB1ADRB3MMEECE1AGTR2
SCHEMBL8920186 0.83 ADRB1 (0.34) ADRB1ADRB3MMEECE1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660840-B1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA GEIGY AG (CH) 1997-05-07 EP disclosed
US-5550119-A ENDOTHELIN-CONVERTING ENZYM INHIBITORS CIBA-GEIGY CORPORATION (US) 1996-08-27 US disclosed
US-5273990-A 5-Phosphonomethyleneamino aryl-substitued alkylene-1H-tetazoles CIBA-GEIGY CORPORATION (US) 1993-12-28 US disclosed