SCHEMBL8924148

SCHEMBL8924148

Clc1cccc(C(OC(c2cccc(Cl)c2)C2CO2)C2CO2)c1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 1/20 0.38
OPRM1 P35372 4/20 0.37
OPRD1 P41143 4/20 0.37
OPRK1 P41145 4/20 0.37
OPRL1 P41146 4/20 0.37
SLC6A4 P31645 9/20 0.37
SLC6A2 P23975 8/20 0.37
SLC6A3 Q01959 4/20 0.37
CYP2D6 P10635 1/20 0.36
ACP3 P15309 1/20 0.36
AOC3 Q16853 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9420774 0.79 SLC6A2 (0.41) HSD17B2OPRM1OPRD1OPRK1OPRL1
SCHEMBL3159928 0.78 SLC6A4 (0.43) SLC6A4SLC6A2SLC6A3
SCHEMBL3687682 0.77 IDO1 (0.44) SLC6A4SLC6A2SLC6A3
SCHEMBL151181 0.77 IDO1 (0.44) SLC6A4SLC6A2SLC6A3
SCHEMBL1357184 0.76 TP53 (0.37)
SCHEMBL11834096 0.76 IDO1 (0.44) OPRM1OPRD1OPRK1OPRL1SLC6A4
Ethylene Glycol SCHEMBL8153345 0.74 CHRM2 (0.38)
SCHEMBL9630636 0.73 GBA1 (0.36)
SCHEMBL11840463 0.72 TP53 (0.42) SLC6A4SLC6A2SLC6A3
SCHEMBL2271173 0.72 SLC6A3 (0.48) SLC6A4SLC6A2SLC6A3AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1254465-C Calcilytic compounds NPS PHARMA INC (US) 2006-05-03 CN disclosed
CN-1221401-A Calcilytic compounds NPS PHARMA INC (US) 1999-06-30 CN disclosed
US-5614518-A Morpholine derivatives as dopamine receptor subtype ligands MERCK SHARP & DOHME LTD. (GB) 1997-03-25 US disclosed
EP-0730593-A1 MORPHOLINE DERIVATIVES AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LTD. (GB) 1996-09-11 EP disclosed
WO-1995014690-A1 MORPHOLINE DERIVATIVES AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1995-06-01 WO disclosed