SCHEMBL8924835

SCHEMBL8924835

CCc1cc(Cl)cc(NC(=S)CCCCc2ccccc2)c1C(=O)OC

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.43
CES1 P23141 4/20 0.41
FAAH O00519 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HSP90AA1 P07900 2/20 0.39
DAGLA Q9Y4D2 1/20 0.39
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
HPGD P15428 2/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HSP90B1 P14625 1/20 0.37
TRPV1 Q8NER1 2/20 0.37
LMNA P02545 1/20 0.37
MGLL Q99685 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8921612 0.82 SMN1; SMN2 (0.37) SMN1; SMN2CES1FAAHKDM4EALDH1A1
SCHEMBL8922395 0.80 CYP4A11 (0.47) SMN1; SMN2ALOX15HPGDALDH1A1LMNA
SCHEMBL8924828 0.80 SMN1; SMN2 (0.43) SMN1; SMN2KDM4EHSP90AA1ALOX15MAPK1
SCHEMBL8921268 0.80 CYP4F2 (0.52) FAAHHPGDALDH1A1
SCHEMBL8783999 0.79 POLB (0.55) SMN1; SMN2KDM4EMAPK1HPGDPOLB
SCHEMBL8920119 0.78 SMN1; SMN2 (0.51) SMN1; SMN2KDM4EALOX15MAPK1HPGD
SCHEMBL8921856 0.76 POLB (0.41) KDM4EHSP90AA1MAPK1POLBALDH1A1
SCHEMBL8921377 0.74 ALDH1A1 (0.46) KDM4EHPGDALDH1A1LMNA
SCHEMBL8921279 0.70 MEN1 (0.40) SMN1; SMN2KDM4EHPGDPOLBALDH1A1
SCHEMBL8921195 0.68 MAPT (0.48) SMN1; SMN2HPGDALDH1A1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633379-A N-METHYLASPARTIC ACID ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-05-27 US disclosed
EP-0685466-A1 3-Heteroaliphatyle-and 3-hetero-(aryle)-aliphatyle-2(1H)-quinolone derivatives CIBA-GEIGY AG (CH) 1995-12-06 EP disclosed