SCHEMBL8925697

SCHEMBL8925697

COC(=O)Cc1c(-c2ccccc2)c(=O)[nH]c2cc(Cl)ccc12

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.58
CYP1A2 P05177 2/20 0.52
POLB P06746 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 1/20 0.52
BLM P54132 1/20 0.52
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CSF1R P07333 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8925137 0.89 ALDH1A1 (0.56) ALDH1A1CYP1A2POLBCYP3A4CYP2C9
SCHEMBL8923670 0.87 KDM4E (0.55) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL8923450 0.82 ALDH1A1 (0.56) ALDH1A1CYP1A2POLBCYP3A4CYP2C9
SCHEMBL8924235 0.81 ALDH1A1 (0.57) ALDH1A1CYP1A2POLBCYP3A4CYP2C9
SCHEMBL8923307 0.80 GPR17 (0.62) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL27554898 0.79 TUBB4A (0.47) ALDH1A1
SCHEMBL8923436 0.79 KDM4E (0.52) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL6701555 0.79 EGFR (0.47) ALDH1A1KDM4E
SCHEMBL28746815 0.78 PTGS2 (0.49)
SCHEMBL8292165 0.78 MCL1 (0.47) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614532-A NERVOUS SYSTEM DISORDERS USING N-METHYLASPARTATE ANTAGONIST MERCK, SHARP & DOHME LTD. (GB) 1997-03-25 US disclosed