SCHEMBL892653

SCHEMBL892653

Cc1ccc(CC(C)N)cc1O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.57
SLC6A2 P23975 3/20 0.57
PNMT P11086 2/20 0.52
ALOX15 P16050 3/20 0.50
ALOX12 P18054 3/20 0.50
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 2/20 0.50
ALDH1A1 P00352 2/20 0.50
ESR1 P03372 2/20 0.50
TP53 P04637 2/20 0.50
CYP3A4 P08684 2/20 0.50
HPGD P15428 2/20 0.50
HTR2A P28223 2/20 0.50
MAPK1 P28482 2/20 0.50
HTR2B P41595 2/20 0.50
RECQL P46063 2/20 0.50
KMT2A Q03164 2/20 0.50
HIF1A Q16665 2/20 0.50
HSD17B10 Q99714 2/20 0.50
SLC6A3 Q01959 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11091077 0.98 TAAR1 (0.55) TAAR1SLC6A2PNMTALOX15ALOX12
SCHEMBL26797474 0.87 ALOX15 (0.53) TAAR1SLC6A2ALOX15ALOX12KDM4E
SCHEMBL11274987 0.85 PLA2G1B (0.47) TAAR1SLC6A2ALOX15ALOX12KDM4E
SCHEMBL633687 0.84 ALOX15 (0.70) TAAR1SLC6A2PNMTALOX15ALOX12
SCHEMBL2562361 0.84 ALOX15 (0.70) TAAR1SLC6A2PNMTALOX15ALOX12
SCHEMBL13660697 0.84 ALOX15 (0.70) TAAR1SLC6A2PNMTALOX15ALOX12
SCHEMBL3960259 0.84 GABRA1 (0.60) SLC6A2ALOX15ALOX12KDM4EMEN1
SCHEMBL29379558 0.84 ALOX15 (0.70) TAAR1SLC6A2PNMTALOX15ALOX12
Bromide SCHEMBL8622617 0.82 ALOX15 (0.68) TAAR1SLC6A2PNMTALOX15ALOX12
SCHEMBL13972055 0.82 PNMT (0.57) TAAR1SLC6A2PNMTHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110294680-A A kind of preparation method in levels Moses spit of fland 北京深蓝海生物医药科技有限公司 2019-10-01 CN claimed
CN-110294680-A A kind of preparation method in levels Moses spit of fland 北京深蓝海生物医药科技有限公司 2019-10-01 CN disclosed
CN-110294680-A A kind of preparation method in levels Moses spit of fland 北京深蓝海生物医药科技有限公司 2019-10-01 CN disclosed
EP-2438819-B9 METHOD FOR PRODUCING A CONCENTRATE OF EICOSAPENTAENOIC AND DOCOSAHEXAENOIC ACID ESTERS GOLDEN OMEGA S A (CL) 2018-05-02 EP disclosed
EP-2438819-B2 METHOD FOR PRODUCING A CONCENTRATE OF EICOSAPENTAENOIC AND DOCOSAHEXAENOIC ACID ESTERS GOLDEN OMEGA S A (CL) 2018-02-14 EP disclosed
US-8981137-B2 Method for producing a concentrate of eicosapentaenoic and docosahexaenoic acids GOLDEN OMEGA S.A. (CL) 2015-03-17 US disclosed
US-20140005425-A1 METHOD FOR PRODUCING A CONCENTRATE OF EICOSAPENTAENOIC AND DOCOSAHEXAENOIC ACIDS GOLDEN OMEGA S.A. (CL) 2014-01-02 US disclosed
US-8586772-B2 Method for producing a concentrate of eicosapentaenoic and docosahexaenoic acid esters GOLDEN OMEGA S.A. (CL) 2013-11-19 US disclosed
EP-2438819-B1 METHOD FOR PRODUCING A CONCENTRATE OF EICOSAPENTAENOIC AND DOCOSAHEXAENOIC ACID ESTERS GOLDEN OMEGA S A (CL) 2013-04-24 EP disclosed
US-20120083616-A1 METHOD FOR PRODUCING A CONCENTRATE OF EICOSAPENTAENOIC AND DOCOSAHEXAENOIC ACID ESTERS GOLDEN OMEGA S.A. (CL) 2012-04-05 US disclosed
US-4824868-A 2-BENZYL-3-SUBSTITUTED-PHENOXYPROPYLAMINES, SEROTONIN UPTAKE INHIBITORS CIBA-GEIGY CORPORATION (US) 1989-04-25 US disclosed
US-4588746-A Propylamine derivatives CIBA-GEIGY CORPORATION (US) 1986-05-13 US disclosed
US-4440940-A HYPOLIPIDEMIC AND ANTIATHEROSCLEROTIC AGENTS AMERICAN CYANAMID COMPANY (US) 1984-04-03 US disclosed
US-4423051-A ANTIATHEROSCLEROTIC AGENTS AND HYPOLIPIDEMIC AGENTS AMERICAN CYANAMID COMPANY (US) 1983-12-27 US disclosed
US-4320137-A Derivatives of perhydro-aza-heterocycles CIBA-GEIGY CORPORATION (US) 1982-03-16 US disclosed
US-4246269-A Antidepressant piperidinones CIBA-GEIGY CORPORATION (US) 1981-01-20 US disclosed
US-4230878-A AND 4-(UNSATURATED ALKYL)AMINOBENZOIC ACIDS AND DERIVATIVES AMERICAN CYANAMID COMPANY (US) 1980-10-28 US disclosed
US-4227014-A ANTILIPEMIC AGENTS, ANTIATHEROSCLEROTIC AGENTS AMERICAN CYANAMID COMPANY (US) 1980-10-07 US disclosed
EP-0003663-A2 Amino-substituted phenyl and heteroaryl compounds, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1979-08-22 EP disclosed
US-4160837-A ANTIDEPRESSANTS CIBA-GEIGY CORPORATION (US) 1979-07-10 US disclosed