SCHEMBL8926780

SCHEMBL8926780

COC(=O)c1ccc(COc2cc(F)ccc2N)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.51
MAOB P27338 1/20 0.50
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
ATM Q13315 1/20 0.43
HSD17B10 Q99714 1/20 0.43
EGFR P00533 1/20 0.42
DPP4 P27487 2/20 0.42
MRGPRX4 Q96LA9 1/20 0.42
PARP1 P09874 1/20 0.42
FFAR4 Q5NUL3 1/20 0.41
PTGER1 P34995 1/20 0.41
GSK3B P49841 1/20 0.41
BACE1 P56817 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8926641 0.82 MAPK14 (0.48) MAPK14MAOBMAPTGAAEGFR
SCHEMBL14157006 0.82 MAPK14 (0.49) MAPK14MAOBKDM4EALDH1A1MAPT
SCHEMBL27698512 0.82 MAPK14 (0.56) MAPK14MAOBPTGER1GSK3BBACE1
SCHEMBL8924125 0.81 ALDH1A1 (0.49) MAPK14MAOBKDM4EALDH1A1MAPT
SCHEMBL14157034 0.79 MAOB (0.53) MAPK14MAOBALDH1A1MAPTGAA
SCHEMBL1457756 0.75 KDM4E (0.61) KDM4EALDH1A1MAPTHPGDGLA
SCHEMBL14156933 0.75 MAOB (0.49) MAPK14MAOBALDH1A1MAPTGAA
SCHEMBL5297104 0.74 MAOB (0.51) MAPK14MAOBMAPTMRGPRX4FFAR4
SCHEMBL1495847 0.74 LOXL2 (0.54) KDM4EALDH1A1MAPTHPGDGLA
Hydrochloric Acid SCHEMBL4418745 0.74 MAPT (0.59) KDM4EALDH1A1MAPTHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639906-A Fluorescent and NMR sensitive pH indicators THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1997-06-17 US disclosed