SCHEMBL8927375

SCHEMBL8927375

CC(=O)Oc1cccc2c(C)c[nH]c12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRPF1 P55201 1/20 0.51
SLC22A6 Q4U2R8 1/20 0.51
KDM4E B2RXH2 5/20 0.48
ALDH1A1 P00352 4/20 0.48
HPGD P15428 4/20 0.48
HTT P42858 3/20 0.46
NR4A2 P43354 1/20 0.44
ACHE P22303 2/20 0.44
PTPN1 P18031 1/20 0.43
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 3/20 0.41
TSHR P16473 2/20 0.41
ESR1 P03372 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
HMGB1 P09429 1/20 0.41
GGT1 P19440 1/20 0.41
PTGS1 P23219 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8927372 0.83 SLC22A6 (0.50) BRPF1SLC22A6KDM4EALDH1A1HPGD
SCHEMBL27728069 0.82 ALDH1A1 (0.44) BRPF1SLC22A6KDM4EALDH1A1HPGD
SCHEMBL9117976 0.81 BRPF1 (0.64) BRPF1SLC22A6KDM4EALDH1A1HPGD
SCHEMBL27961376 0.79 ALDH1A1 (0.61) BRPF1SLC22A6KDM4EALDH1A1HPGD
SCHEMBL27858183 0.78 KDM4E (0.39) BRPF1SLC22A6KDM4EALDH1A1HPGD
SCHEMBL8926562 0.78 HTR2A (0.57) BRPF1KDM4EALDH1A1HPGDHTT
SCHEMBL27612163 0.76 SOS2 (0.60) SLC22A6ACHEMTNR1AMTNR1B
SCHEMBL28034293 0.75 SLC22A6 (0.61) BRPF1SLC22A6KDM4EALDH1A1HPGD
SCHEMBL30630330 0.75 HTR6 (0.70) ACHEMTNR1AMTNR1B
SCHEMBL27085080 0.75 HTR6 (0.70) ACHEMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101040037-B Organic compounds GIVAUDAN SA 2010-08-18 CN disclosed
CN-101040037-A Organic compounds GIVAUDAN SA (CH) 2007-09-19 CN disclosed
US-5614498-A OLIGOPEPTIDES, BRONCHDILATORS BANYU PHARMACEUTICAL CO., LTD. (JP) 1997-03-25 US disclosed
US-5496928-A Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
EP-0555537-A2 Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-18 EP disclosed