SCHEMBL8927900

SCHEMBL8927900

CC1CN(C(=O)O)CCN(C(=O)O)CCN(CC(O)C(F)(F)F)CCN1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
MEN1 O00255 1/20 0.37
PDK1 Q15118 2/20 0.34
PDK2 Q15119 2/20 0.34
PDK3 Q15120 2/20 0.34
PDK4 Q16654 2/20 0.34
PIK3CD O00329 1/20 0.32
TAAR1 Q96RJ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928194 0.90 PDK1 (0.35) KMT2ALMNAHTTPDK1PDK2
SCHEMBL8302334 0.84 PIK3CD (0.38) LMNAHTTPIK3CD
SCHEMBL13505787 0.83 KMT2A (0.58) KMT2ALMNAHTTMEN1PIK3CD
SCHEMBL5551312 0.81 KDM4E (0.43) KMT2ALMNAMEN1PIK3CD
SCHEMBL5551323 0.81 PIK3CD (0.33) LMNAPIK3CD
SCHEMBL8560245 0.80 ALDH1A1 (0.43) KMT2AHTTMEN1
SCHEMBL4150920 0.78 TSHR (0.41) LMNAHTTPDK1PDK2PDK3
SCHEMBL7995036 0.78 TSHR (0.41) LMNAHTTPDK1PDK2PDK3
SCHEMBL8559141 0.78 ALDH1A1 (0.52) KMT2ALMNAHTTMEN1
SCHEMBL8927884 0.77 PDK1 (0.41) PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5690909-A USEFUL AS NMR AND X-RAY DIAGNOSTIC AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 1997-11-25 US disclosed
EP-0700393-B1 MACROCYCLIC METAL COMPLEXES CONTAINING FLUORINE SCHERING AG (DE) 1997-10-22 EP disclosed
EP-0700393-A1 MACROCYCLIC METAL COMPLEXES CONTAINING FLUORINE SCHERING AG (DE) 1996-03-13 EP disclosed
WO-1994027978-A1 MACROCYCLIC METAL COMPLEXES CONTAINING FLUORINE SCHERING AKTIENGESELLSCHAFT (DE) 1994-12-08 WO disclosed