SCHEMBL8928248

SCHEMBL8928248

CCOC(=O)C1=C(C)NC(C)=C(C#N)C1c1cccc(-n2cncn2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 7/20 0.49
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C9 P11712 3/20 0.47
CYP2C19 P33261 3/20 0.47
MAPT P10636 3/20 0.46
ALDH1A1 P00352 2/20 0.46
CACNA1F O60840 4/20 0.46
CACNA1D Q01668 4/20 0.46
CACNA1S Q13698 4/20 0.46
ADORA3 P0DMS8 2/20 0.46
HIF1A Q16665 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
MAPK1 P28482 1/20 0.43
GPR55 Q9Y2T6 1/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928269 0.85 SMN1; SMN2 (0.46) MAPTALDH1A1MEN1KMT2ALMNA
SCHEMBL8928277 0.84 CACNA1C (0.54) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6137184 0.79 CACNA1C (0.64) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7586726 0.78 CACNA1C (0.60) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7586763 0.76 CACNA1C (0.60) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7590982 0.75 CACNA1F (0.80) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7588425 0.73 ABCC1 (0.57) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8928255 0.73 CHRNA7 (0.44) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL7269131 0.73 CACNA1F (0.54) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL30357940 0.73 CACNA1F (0.54) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP claimed
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP disclosed