SCHEMBL8928255

SCHEMBL8928255

CC1=C(C#N)C(c2cccc(-n3cncn3)c2)C(C#N)=C(C)N1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.44
MET P08581 1/20 0.38
CYP2A6 P11509 1/20 0.37
ALDH1A1 P00352 4/20 0.33
MAPT P10636 3/20 0.33
KMT2A Q03164 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
MEN1 O00255 2/20 0.33
CYP2D6 P10635 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
DPP4 P27487 1/20 0.32
ADORA3 P0DMS8 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928269 0.86 SMN1; SMN2 (0.46) CHRNA7METCYP2A6ALDH1A1MAPT
SCHEMBL8928246 0.79 IDO1 (0.44) METCYP2A6MAPTCYP1A2CYP3A4
SCHEMBL8928248 0.73 CACNA1C (0.49) ALDH1A1MAPTKMT2ACYP1A2CYP3A4
SCHEMBL13295965 0.71 CUL4A (0.53) METALDH1A1MAPTKMT2ACYP1A2
SCHEMBL27965992 0.70 GRM5 (0.51) CYP2A6ALDH1A1KDM4EADORA3SMN1; SMN2
SCHEMBL13295967 0.70 ALDH1A1 (0.53) ALDH1A1MAPTKMT2AKDM4EHPGD
SCHEMBL11926858 0.69 CYP2A6 (0.62) CHRNA7CYP2A6ALDH1A1CYP1A2CYP3A4
SCHEMBL4442073 0.69 KMO (0.41) METALDH1A1MAPTKMT2ACYP1A2
SCHEMBL9454459 0.68 CYP2A6 (0.53) CHRNA7CYP2A6ALDH1A1KMT2ACYP1A2
SCHEMBL8928234 0.67 GRK6 (0.43) CHRNA7CYP2A6ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP claimed
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP disclosed