SCHEMBL8928277

SCHEMBL8928277

CCOC(=O)C1=C(C)NC(C)=C(C#N)C1c1cccc(-n2ccnc2)c1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 6/20 0.54
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
CACNA1F O60840 3/20 0.46
CACNA1D Q01668 3/20 0.46
CACNA1S Q13698 3/20 0.46
ADORA3 P0DMS8 2/20 0.46
NR3C2 P08235 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269131 0.91 CACNA1F (0.54) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL30357940 0.91 CACNA1F (0.54) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8928241 0.88 KDM4E (0.53) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8928204 0.88 CACNA1C (0.40) CACNA1CALDH1A1MAPT
SCHEMBL7277695 0.88 CACNA1C (0.48) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7275109 0.87 ADORA3 (0.59) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8860432 0.85 POLB (0.49) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL8928281 0.84 POLB (0.48) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL8928248 0.84 CACNA1C (0.49) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10475638 0.80 CACNA1F (0.50) CACNA1CCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP claimed
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP disclosed