SCHEMBL8928378

SCHEMBL8928378

CCc1cc2c(s1)-n1c(Br)nnc1CN=C2c1ccccc1Cl

nearest known ligand 0.79

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.79
PDE4D Q08499 1/20 0.79
PTAFR P25105 17/20 0.62
TDP1 Q9NUW8 1/20 0.58
CYP3A4 P08684 1/20 0.53
ALOX15 P16050 1/20 0.53
GABRA1 P14867 1/20 0.52
TSHR P16473 1/20 0.52
GABRA5 P31644 1/20 0.52
GABRA3 P34903 1/20 0.52
GABRA2 P47869 1/20 0.52
GABRB2 P47870 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10511151 0.92 OPRK1 (0.67) OPRK1PDE4DPTAFRTDP1CYP3A4
SCHEMBL8928481 0.90 OPRK1 (0.84) OPRK1PDE4DPTAFRCYP3A4ALOX15
Etizolam SCHEMBL42920 0.88 OPRK1 (1.00) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928449 0.88 OPRK1 (0.80) OPRK1PDE4DPTAFRCYP3A4ALOX15
Etizolam SCHEMBL30665015 0.88 OPRK1 (1.00) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928568 0.85 OPRK1 (0.76) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928839 0.85 OPRK1 (0.76) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928541 0.85 OPRK1 (0.76) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8878112 0.85 OPRK1 (0.79) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928415 0.85 OPRK1 (0.74) OPRK1PDE4DPTAFRCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776892-A1 THIENYLAZOLE COMPOUND AND THIENOTRIAZOLODIAZEPINE COMPOUND YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-06-04 EP disclosed