SCHEMBL8928416

SCHEMBL8928416

CCc1cc2c(s1)-n1c(nnc1CNC(=O)c1cc3cc(OC)ccc3[nH]1)CN=C2c1ccccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.53
PDE4D Q08499 1/20 0.53
KDM4E B2RXH2 7/20 0.46
MAPT P10636 4/20 0.46
ALDH1A1 P00352 3/20 0.46
PTAFR P25105 7/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
DRD4 P21917 1/20 0.41
PLCG2 P16885 1/20 0.41
HTR2A P28223 1/20 0.41
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928615 0.92 OPRK1 (0.55) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928421 0.92 OPRK1 (0.57) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928499 0.91 OPRK1 (0.53) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928523 0.86 PTAFR (0.49) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928639 0.84 OPRK1 (0.55) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928487 0.84 OPRK1 (0.46) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928590 0.83 OPRK1 (0.46) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928848 0.83 OPRK1 (0.44) OPRK1PDE4DKDM4EALDH1A1DRD2
SCHEMBL8929052 0.82 OPRK1 (0.58) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928420 0.82 OPRK1 (0.59) OPRK1PDE4DPTAFRCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776892-A1 THIENYLAZOLE COMPOUND AND THIENOTRIAZOLODIAZEPINE COMPOUND YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-06-04 EP disclosed