SCHEMBL8930663

SCHEMBL8930663

CC1(C)Oc2cc3c(c(C(O)(c4c5c(cc6c4OC(C)(C)O6)OC(C)(C)O5)c4c5c(cc6c4OC(C)(C)O6)OC(C)(C)O5)c2O1)OC(C)(C)O3

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050476 0.82 TSHR (0.35) TSHR
SCHEMBL7523102 0.82 TSHR (0.35) TSHR
SCHEMBL9719308 0.73 TSHR (0.62) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8930654 0.72
SCHEMBL7519328 0.71 TSHR (1.00) TSHRCYP1A2CYP2C9CYP2C19
SCHEMBL8930700 0.71 TSHR (0.52) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8930686 0.70 TSHR (0.56) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8930698 0.69
SCHEMBL27382503 0.68 TSHR (0.38) TSHR
SCHEMBL12412424 0.66 TSHR (0.45) TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0423482-B1 5H-furan-2-one derivatives BAYER AG (DE) 1995-01-11 EP claimed
US-5599522-A CONTRAST ENHANCING AGENTS NYCOMED IMAGING AS (NO) 1997-02-04 US disclosed
EP-0515458-B1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI NYCOMED INNOVATION AB (SE) 1995-08-23 EP disclosed
EP-0515458-A1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI. HAFSLUND NYCOMED INNOVATION (SE) 1992-12-02 EP disclosed
WO-1991012024-A1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI HAFSLUND NYCOMED INNOVATION AB (SE) 1991-08-22 WO disclosed