SCHEMBL8931355

SCHEMBL8931355

CCC(=O)Nc1ccc2[nH]c(C)c(CCN(C)Cc3cncc(C(=O)NO)n3)c2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 1/20 0.48
ALDH1A1 P00352 6/20 0.40
HPGD P15428 2/20 0.40
MAPT P10636 10/20 0.39
NPSR1 Q6W5P4 4/20 0.39
LMNA P02545 4/20 0.39
KMT2A Q03164 6/20 0.38
KDM4E B2RXH2 1/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 4/20 0.37
GAA P10253 1/20 0.37
EPHB2 P29323 1/20 0.37
TERT O14746 1/20 0.36
MAPK1 P28482 1/20 0.36
PDE10A Q9Y233 1/20 0.36
ATM Q13315 2/20 0.36
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8181328 0.86 HTR1F (0.47) HTR1FALDH1A1HPGDMAPTNPSR1
SCHEMBL8931383 0.85 ALDH1A1 (0.41) HTR1FALDH1A1HPGDMAPTKMT2A
SCHEMBL7139743 0.77 HTR1F (0.68) HTR1FALDH1A1HPGDMAPTNPSR1
SCHEMBL8181303 0.71 ALDH1A1 (0.43) HTR1FALDH1A1HPGDMAPTKMT2A
SCHEMBL8181951 0.70 CNR1 (0.49) HTR1FALDH1A1HPGDKMT2AKDM4E
SCHEMBL7141203 0.69 HTR1F (0.73) HTR1FALDH1A1MAPTNPSR1LMNA
Benzoic Acid SCHEMBL8191205 0.69 HTR1F (0.45) HTR1FALDH1A1HPGDMAPTNPSR1
SCHEMBL7144771 0.69 HTR1F (0.83) HTR1FALDH1A1HPGDMAPTNPSR1
SCHEMBL8598857 0.68 HTR1F (0.81) HTR1FALDH1A1HPGDMAPTNPSR1
SCHEMBL7140886 0.68 HTR1F (0.60) HTR1FALDH1A1MAPTKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997013512-A1 N-[2-SUBSTITUTED-3-(2-AMINOETHYL)-1H-INDOL-5-YL]-AMIDES: NEW 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1997-04-17 WO disclosed