SCHEMBL8933090

SCHEMBL8933090

CC(C)(C)OC(=O)C=NCC(=O)N1CCC[C@]1(C(=O)O)C1CCCCC1.N#Cc1ccc(C(N)=O)cn1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.35
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
CPT2 P23786 1/20 0.31
CPT1A P50416 1/20 0.31
OPRM1 P35372 2/20 0.31
OPRK1 P41145 2/20 0.31
TACR3 P29371 1/20 0.30
OPRD1 P41143 1/20 0.30
CHEK2 O96017 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8725915 0.88 OPRM1 (0.30) OPRM1OPRK1
SCHEMBL8933077 0.85
SCHEMBL6477215 0.85 JAK2 (0.37) GPR119JAK2JAK1CTSSCTSK
SCHEMBL6476534 0.85 JAK2 (0.36) GPR119JAK2JAK1CTSSCTSK
SCHEMBL6477307 0.82 CTSS (0.34) JAK2JAK1CTSSCTSKCPT2
SCHEMBL8933278 0.79 OPRK1 (0.32) OPRK1
SCHEMBL8722615 0.77 HRH3 (0.34) OPRK1
SCHEMBL8725919 0.77
SCHEMBL6489531 0.74 NPFFR1 (0.35) OPRM1OPRK1OPRD1
SCHEMBL8722553 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996025426-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1996-08-22 WO disclosed