SCHEMBL8933482

SCHEMBL8933482

N#Cc1ccc2c(c1)C(c1ccccc1F)=NCc1nccn1-2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.50
GABRA5 P31644 4/20 0.50
GABRA2 P47869 4/20 0.50
GABRB2 P47870 2/20 0.50
PTAFR P25105 10/20 0.48
GABRA3 P34903 5/20 0.47
GABRG2 P18507 3/20 0.45
GABRB3 P28472 3/20 0.45
SLC22A1 O15245 1/20 0.40
ABCB11 O95342 1/20 0.40
CYP3A4 P08684 1/20 0.40
DRD3 P35462 1/20 0.40
OPRK1 P41145 1/20 0.40
PDE4D Q08499 1/20 0.40
CCNE2 O96020 1/20 0.39
EGFR P00533 1/20 0.39
CDK1 P06493 1/20 0.39
CDK4 P11802 1/20 0.39
SRC P12931 1/20 0.39
CCND1 P24385 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11825305 0.87 GABRA1 (0.51) GABRA1GABRA5GABRA2GABRB2PTAFR
SCHEMBL11830483 0.85 GABRA1 (0.58) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL11826943 0.85 PTAFR (0.47) GABRA1GABRA5GABRA2GABRB2PTAFR
SCHEMBL11830831 0.83 GABRA1 (0.49) GABRA1GABRA5GABRA2GABRB2PTAFR
SCHEMBL32673434 0.83 OPRK1 (0.57) GABRA1GABRA5GABRA2PTAFRGABRA3
SCHEMBL11729005 0.83 OPRK1 (0.57) GABRA1GABRA5GABRA2PTAFRGABRA3
SCHEMBL11827953 0.81 GABRA1 (0.53) GABRA1GABRA5GABRA2GABRB2PTAFR
SCHEMBL8933572 0.80 CYP3A4 (0.47) GABRA1GABRA5GABRA2GABRB2PTAFR
SCHEMBL11835141 0.80 PTAFR (0.45) GABRA1GABRA5GABRA2GABRB2PTAFR
SCHEMBL11826404 0.79 GABRA3 (0.63) GABRA1GABRA5GABRA2GABRB2PTAFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996023790-A1 ACETYLIMIDAZOBENZODIAZEPINES F. HOFFMANN-LA ROCHE AG (CH) 1996-08-08 WO disclosed
US-3933794-A CENTRAL NERVOUS SYSTEM DEPRESSANTS THE UPJOHN COMPANY (US) 1976-01-20 US disclosed