SCHEMBL8933625

SCHEMBL8933625

N#Cc1ccc2c(c1)C(c1ccccc1F)=NCC(=S)N2

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 11/20 0.69
CCNE2 O96020 1/20 0.56
EGFR P00533 1/20 0.56
CDK1 P06493 1/20 0.56
CDK4 P11802 1/20 0.56
SRC P12931 1/20 0.56
CCND1 P24385 1/20 0.56
CCNE1 P24864 1/20 0.56
CDK2 P24941 1/20 0.56
KDR P35968 1/20 0.56
CCNA1 P78396 1/20 0.56
PTK2 Q05397 1/20 0.56
ALOX12 P18054 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
GABRA1 P14867 3/20 0.50
GABRA5 P31644 3/20 0.50
GABRA2 P47869 3/20 0.50
GABRB2 P47870 3/20 0.50
GABRA3 P34903 2/20 0.50
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10404819 0.86 ALOX12 (0.72) CHRM1CCNE2EGFRCDK1CDK4
SCHEMBL7320239 0.86 GABRA1 (0.69) CHRM1CCNE2EGFRCDK1CDK4
SCHEMBL7321076 0.84 CHRM1 (0.67) CHRM1CCNE2EGFRCDK1CDK4
SCHEMBL7324382 0.84 CHRM1 (0.77) CHRM1CCNE2CCNE1CDK2ALOX12
SCHEMBL11733109 0.82 CHRM1 (0.73) CHRM1CCNE2CCNE1CDK2ALOX12
SCHEMBL30320323 0.81 CHRM1 (1.00) CHRM1CCNE2CCNE1CDK2ALOX12
SCHEMBL7324283 0.81 CHRM1 (0.73) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL7950385 0.81 CHRM1 (1.00) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5
SCHEMBL7328311 0.81 CHRM1 (1.00) CHRM1CCNE2CCNE1CDK2ALOX12
SCHEMBL11825759 0.80 CHRM1 (0.74) CHRM1ALOX12SMN1; SMN2GABRA1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996023790-A1 ACETYLIMIDAZOBENZODIAZEPINES F. HOFFMANN-LA ROCHE AG (CH) 1996-08-08 WO disclosed
US-3933794-A CENTRAL NERVOUS SYSTEM DEPRESSANTS THE UPJOHN COMPANY (US) 1976-01-20 US disclosed